1a8t
From PDBWiki
METALLO-BETA-LACTAMASE IN COMPLEX WITH L-159,061
| Authors | Toney, J.H. Fitzgerald, P.M. Grover-Sharma, N. Olson, S.H. May, W.J. Sundelof, J.G. Vanderwall, D.E. Cleary, K.A. Grant, S.K. Wu, J.K. Kozarich, J.W. Pompliano, D.L. Hammond, G.G. |
| Citation | Antibiotic sensitization using biphenyl tetrazoles as potent inhibitors of Bacteroides fragilis metallo-beta-lactamase. |
| Release date | 1998-10-14 |
| Exp. Method | X-RAY DIFFRACTION |
| Resolution | 2.55 Å |
| Classification | HYDROLASE |
Sequence
Chain A (232 residues): Blast Uniprot EC 3.5.2.6AQKSVKISDDISITQLSDKVYTYVSLAEIEGWGMVPSNGMIVINNHQAALLDTPINDAQTEMLVNWVTDSLHAKVTTFIP NHWHGDCIGGLGYLQRKGVQSYANQMTIDLAKEKGLPVPEHGFTDSLTVSLDGMPLQCYYLGGGHATDNIVVWLPTENIL FGGCMLKDNQTTSIGNISDADVTAWPKTLDKVKAKFPSARYVVPGHGNYGGTELIEHTKQIVNQYIESTSKPChain B (232 residues): Blast Uniprot EC 3.5.2.6
AQKSVKISDDISITQLSDKVYTYVSLAEIEGWGMVPSNGMIVINNHQAALLDTPINDAQTEMLVNWVTDSLHAKVTTFIP NHWHGDCIGGLGYLQRKGVQSYANQMTIDLAKEKGLPVPEHGFTDSLTVSLDGMPLQCYYLGGGHATDNIVVWLPTENIL FGGCMLKDNQTTSIGNISDADVTAWPKTLDKVKAKFPSARYVVPGHGNYGGTELIEHTKQIVNQYIESTSKP
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