1a9u
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THE COMPLEX STRUCTURE OF THE MAP KINASE P38/SB203580
| Authors | Wang, Z. Canagarajah, B.J. Boehm, J.C. Kassisa, S. Cobb, M.H. Young, P.R. Abdel-Meguid, S. Adams, J.L. Goldsmith, E.J. |
| Citation | Structural basis of inhibitor selectivity in MAP kinases. |
| Release date | 2003-04-01 |
| Exp. Method | X-RAY DIFFRACTION |
| Resolution | 2.5 Å |
| Classification | TRANSFERASE |
Sequence
Chain A (379 residues): Blast Uniprot EC 2.7.11.24GSSHHHHHHSSGLVPRGSHMSQERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQS IIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYI HSADIIHRDLKPSNLAVNEDCELKILDFGLARHTDDEMTGYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRT LFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQ ALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPPLDQEEMES
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| Databases | Visualization tools | Analysis tools | Quarternary structure |
|---|---|---|---|
Categories: A9 | PDB entry | X-RAY DIFFRACTION | TRANSFERASE | HOMO SAPIENS | 2003 | EC 2.7.11.24

