1a9u

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1a9u

THE COMPLEX STRUCTURE OF THE MAP KINASE P38/SB203580

Authors Wang, Z. Canagarajah, B.J. Boehm, J.C. Kassisa, S. Cobb, M.H. Young, P.R. Abdel-Meguid, S. Adams, J.L. Goldsmith, E.J.
Citation Structural basis of inhibitor selectivity in MAP kinases.
Release date 2003-04-01
Exp. Method X-RAY DIFFRACTION
Resolution 2.5 Å
Classification TRANSFERASE

Sequence

Chain A (379 residues): Blast Uniprot EC 2.7.11.24
GSSHHHHHHSSGLVPRGSHMSQERPTFYRQELNKTIWEVPERYQNLSPVGSGAYGSVCAAFDTKTGLRVAVKKLSRPFQS
IIHAKRTYRELRLLKHMKHENVIGLLDVFTPARSLEEFNDVYLVTHLMGADLNNIVKCQKLTDDHVQFLIYQILRGLKYI
HSADIIHRDLKPSNLAVNEDCELKILDFGLARHTDDEMTGYVATRWYRAPEIMLNWMHYNQTVDIWSVGCIMAELLTGRT
LFPGTDHIDQLKLILRLVGTPGAELLKKISSESARNYIQSLTQMPKMNFANVFIGANPLAVDLLEKMLVLDSDKRITAAQ
ALAHAYFAQYHDPDDEPVADPYDQSFESRDLLIDEWKSLTYDEVISFVPPPLDQEEMES


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