1eb2

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TRYPSIN INHIBITOR COMPLEX (BPO)

Authors Liebeschuetz, J.W. Jones, S.D. Morgan, P.J. Murray, C.W. Rimmer, A.D. Roscoe, J.M.E. Waszkowycz, B. Welsh, P.M. Wylie, W.A. Young, S.C. Martin, H. Mahler, J. Brady, R.L. Wilkinson, K.W.
Citation Pro_Select: Combining Structure-Based Drug Design and Array-Based Chemistry for Rapid Lead Discovery. 2. The Development of a Series of Highly Potent and Selective Factor Xa Inhibitors PubMed
Release date 2002-02-11
Exp. Method X-RAY DIFFRACTION
Resolution 2.0 Å
Classification HYDROLASE

Sequence

Chain(s) A (223 residues): Blast EC 3.4.21.4
IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNT
LNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNM
FCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN

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