1eb2
From PDBWiki
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TRYPSIN INHIBITOR COMPLEX (BPO)
| Authors | Liebeschuetz, J.W. Jones, S.D. Morgan, P.J. Murray, C.W. Rimmer, A.D. Roscoe, J.M.E. Waszkowycz, B. Welsh, P.M. Wylie, W.A. Young, S.C. Martin, H. Mahler, J. Brady, R.L. Wilkinson, K.W. |
| Citation | Pro_Select: Combining Structure-Based Drug Design and Array-Based Chemistry for Rapid Lead Discovery. 2. The Development of a Series of Highly Potent and Selective Factor Xa Inhibitors PubMed |
| Release date | 2002-02-11 |
| Exp. Method | X-RAY DIFFRACTION |
| Resolution | 2.0 Å |
| Classification | HYDROLASE |
Sequence
Chain(s) A (223 residues): Blast EC 3.4.21.4IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNT LNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNM FCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN
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