1gfz
From PDBWiki
FLAVOPIRIDOL INHIBITS GLYCOGEN PHOSPHORYLASE BY BINDING AT THE INHIBITOR SITE
| Authors | Oikonomakos, N.G. Schnier, J.B. Zographos, S.E. Skamnaki, V.T. Tsitsanou, K.E. Johnson, L.N. |
| Citation | Flavopiridol inhibits glycogen phosphorylase by binding at the inhibitor site. |
| Release date | 2002-06-14 |
| Exp. Method | X-RAY DIFFRACTION |
| Resolution | 2.3 Å |
| Classification | TRANSFERASE |
Sequence
Chain A (842 residues): Blast Uniprot EC 2.4.1.1SRPLSDQEKRKQISVRGLAGVENVTELKKNFNRHLHFTLVKDRNVATPRDYYFALAHTVRDHLVGRWIRTQQHYYEKDPK RIYYLSLEFYMGRTLQNTMVNLALENACDEATYQLGLDMEELEEIEEDAGLGNGGLGRLAACFLDSMATLGLAAYGYGIR YEFGIFNQKICGGWQMEEADDWLRYGNPWEKARPEFTLPVHFYGRVEHTSQGAKWVDTQVVLAMPYDTPVPGYRNNVVNT MRLWSAKAPNDFNLKDFNVGGYIQAVLDRNLAENISRVLYPNDNFFEGKELRLKQEYFVVAATLQDIIRRFKSSKFGCRD PVRTNFDAFPDKVAIQLNDTHPSLAIPELMRVLVDLERLDWDKAWEVTVKTCAYTNHTVIPEALERWPVHLLETLLPRHL QIIYEINQRFLNRVAAAFPGDVDRLRRMSLVEEGAVKRINMAHLCIAGSHAVNGVARIHSEILKKTIFKDFYELEPHKFQ NKTNGITPRRWLVLCNPGLAEIIAERIGEEYISDLDQLRKLLSYVDDEAFIRDVAKVKQENKLKFAAYLEREYKVHINPN SLFDVQVKRIHEYKRQLLNCLHVITLYNRIKKEPNKFVVPRTVMIGGKAAPGYHMAKMIIKLITAIGDVVNHDPVVGDRL RVIFLENYRVSLAEKVIPAADLSEQISTAGTEASGTGNMKFMLNGALTIGTMDGANVEMAEEAGEENFFIFGMRVEDVDR LDQRGYNAQEYYDRIPELRQIIEQLSSGFFSPKQPDLFKDIVNMLMHHDRFKVFADYEEYVKCQERVSALYKNPREWTRM VIRNIATSGKFSSDRTIAQYAREIWGVEPSRQRLPAPDEKIP
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| Databases | Visualization tools | Analysis tools | Quarternary structure |
|---|---|---|---|
Categories: GF | PDB entry | X-RAY DIFFRACTION | TRANSFERASE | 2002 | EC 2.4.1.1

