1gj6

From PDBWiki

Jump to: navigation, search
1gj6

ENGINEERING INHIBITORS HIGHLY SELECTIVE FOR THE S1 SITES OF SER190 TRYPSIN-LIKE SERINE PROTEASE DRUG TARGETS

Authors Katz, B.A. Sprengeler, P.A. Luong, C. Verner, E. Elrod, K. Kirtley, M. Janc, J. Spencer, J.R. Breitenbucher, J.G. Hui, H. McGee, D. Allen, D. Martelli, A. Mackman, R.L.
Citation Engineering inhibitors highly selective for the S1 sites of Ser190 trypsin-like serine protease drug targets. PubMed
Release date 2002-04-27
Exp. Method X-RAY DIFFRACTION
Resolution 1.5 Å
Classification hydrolase

Sequence

Chain A (223 residues): Blast Uniprot EC 3.4.21.4
IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNT
LNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNM
FCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN


User comments


Links

 Search for 1gj6 in:

Databases Visualization tools Analysis tools Quarternary structure
Personal tools