1gj6
From PDBWiki
ENGINEERING INHIBITORS HIGHLY SELECTIVE FOR THE S1 SITES OF SER190 TRYPSIN-LIKE SERINE PROTEASE DRUG TARGETS
| Authors | Katz, B.A. Sprengeler, P.A. Luong, C. Verner, E. Elrod, K. Kirtley, M. Janc, J. Spencer, J.R. Breitenbucher, J.G. Hui, H. McGee, D. Allen, D. Martelli, A. Mackman, R.L. |
| Citation | Engineering inhibitors highly selective for the S1 sites of Ser190 trypsin-like serine protease drug targets. PubMed |
| Release date | 2002-04-27 |
| Exp. Method | X-RAY DIFFRACTION |
| Resolution | 1.5 Å |
| Classification | hydrolase |
Sequence
Chain A (223 residues): Blast Uniprot EC 3.4.21.4IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNT LNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNM FCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN
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| Databases | Visualization tools | Analysis tools | Quarternary structure |
|---|---|---|---|
Categories: GJ | PDB entry | X-RAY DIFFRACTION | HYDROLASE | 2002 | EC 3.4.21.4

