1gkd

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1gkd

MMP9 ACTIVE SITE MUTANT-INHIBITOR COMPLEX

Authors Rowsell, S. Hawtin, P. Minshull, C.A. Jepson, H. Brockbank, S.M. Barratt, D.G. Slater, A.M. McPheat, W.L. Waterson, D. Henney, A.M. Pauptit, R.A.
Citation Crystal structure of human MMP9 in complex with a reverse hydroxamate inhibitor. PubMed
Release date 2003-04-01
Exp. Method X-RAY DIFFRACTION
Resolution 2.1 Å
Classification HYDROLASE

Sequence

Chain A (163 residues): Blast Uniprot
MFQTFEGDLKWHHHNITYWIQNYSEDLPRAVIDDAFARAFALWSAVTPLTFTRVYSRDADIVIQFGVAEHGDGYPFDGKD
GLLAHAFPPGPGIQGDAHFDDDELWSLGKGQGYSLFLVAAHQFGHALGLDHSSVPEALMYPMYRFTEGPPLHKDDVNGIR
HLY
Chain B (163 residues): Blast Uniprot
MFQTFEGDLKWHHHNITYWIQNYSEDLPRAVIDDAFARAFALWSAVTPLTFTRVYSRDADIVIQFGVAEHGDGYPFDGKD
GLLAHAFPPGPGIQGDAHFDDDELWSLGKGQGYSLFLVAAHQFGHALGLDHSSVPEALMYPMYRFTEGPPLHKDDVNGIR
HLY


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