1hj1

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1hj1

RAT OESTROGEN RECEPTOR BETA LIGAND-BINDING DOMAIN IN COMPLEX WITH PURE ANTIOESTROGEN ICI164,384

Authors Pike, A.C. Brzozowski, A.M. Walton, J. Hubbard, R.E. Thorsell, A.G. Li, Y.L. Gustafsson, J.A. Carlquist, M.
Citation Structural insights into the mode of action of a pure antiestrogen.
Release date 2002-01-04
Exp. Method X-RAY DIFFRACTION
Resolution 2.3 Å
Classification NUCLEAR RECEPTOR

Sequence

Chain A (255 residues): Blast Uniprot
VKELLLSTLSPEQLVLTLLEAEPPNVLVSRPSMPFTEASMMMSLTKLADKELVHMIGWAKKIPGFVELSLLDQVRLLESC
WMEVLMVGLMWRSIDHPGKLIFAPDLVLDRDEGKCVEGILEIFDMLLATTSRFRELKLQHKEYLCVKAMILLNSSMYPLA
SANQEAESSRKLTHLLNAVTDALVWVIAKSGISSQQQSVRLANLLMLLSHVRHISNKGMEHLLSMKCKNVVPVYDLLLEM
LNAHLTRGYKSSISG


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