1jin

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1jin

P450eryF/ketoconazole

Authors Cupp-Vickery, J.R. Garcia, C. Hofacre, A. McGee-Estrada, K.
Citation Ketoconazole-induced conformational changes in the active site of cytochrome P450eryF. PubMed
Release date 2001-10-17
Exp. Method X-RAY DIFFRACTION
Resolution 2.3 Å
Classification HYDROLASE

Sequence

Chain A (403 residues): Blast Uniprot EC 1.-.-.-
ATVPDLESDSFHVDWYSTYAELRETAPVTPVRFLGQDAWLVTGYDEAKAALSDLRLSSDPKKKYPGVEVEFPAYLGFPED
VRNYFATNMGTSDPPTHTRLRKLVSQEFTVRRVEAMRPRVEQITAELLDEVGDSGVVDIVDRFAHPLPIKVICELLGVDE
AARGAFGRWSSEILVMDPERAEQRGQAAREVVNFILDLVERRRTEPGDDLLSALISVQDDDDGRLSADELTSIALVLLLA
GFEASVSLIGIGTYLLLTHPDQLALVRADPSALPNAVEEILRYIAPPETTTRFAAEEVEIGGVAIPQYSTVLVANGAANR
DPSQFPDPHRFDVTRDTRGHLSFGQGIHFCMGRPLAKLEGEVALRALFGRFPALSLGIDADDVVWRRSLLLRGIDHLPVR
LDG


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