1jip
From PDBWiki
P450eryF(A245S)/ketoconazole
| Authors | Cupp-Vickery, J.R. Garcia, C. Hofacre, A. McGee-Estrada, K. |
| Citation | Ketoconazole-induced conformational changes in the active site of cytochrome P450eryF. PubMed |
| Release date | 2001-10-17 |
| Exp. Method | X-RAY DIFFRACTION |
| Resolution | 2.0 Å |
| Classification | HYDROLASE |
Sequence
Chain A (403 residues): Blast Uniprot EC 1.-.-.-TTVPDLESDSFHVDWYRTYAELRETAPVTPVRFLGQDAWLVTGYDEAKAALSDLRLSSDPKKKYPGVEVEFPAYLGFPED VRNYFATNMGTSDPPTHTRLRKLVSQEFTVRRVEAMRPRVEQITAELLDEVGDSGVVDIVDRFAHPLPIKVICELLGVDE KYRGEFGRWSSEILVMDPERAEQRGQAAREVVNFILDLVERRRTEPGDDLLSALIRVQDDDDGRLSADELTSIALVLLLA GFESSVSLIGIGTYLLLTHPDQLALVRRDPSALPNAVEEILRYIAPPETTTRFAAEEVEIGGVAIPQYSTVLVANGAANR DPKQFPDPHRFDVTRDTRGHLSFGQGIHFCMGRPLAKLEGEVALRALFGRFPALSLGIDADDVVWRRSLLLRGIDHLPVR LDG
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