1jip

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1jip

P450eryF(A245S)/ketoconazole

Authors Cupp-Vickery, J.R. Garcia, C. Hofacre, A. McGee-Estrada, K.
Citation Ketoconazole-induced conformational changes in the active site of cytochrome P450eryF. PubMed
Release date 2001-10-17
Exp. Method X-RAY DIFFRACTION
Resolution 2.0 Å
Classification HYDROLASE

Sequence

Chain A (403 residues): Blast Uniprot EC 1.-.-.-
TTVPDLESDSFHVDWYRTYAELRETAPVTPVRFLGQDAWLVTGYDEAKAALSDLRLSSDPKKKYPGVEVEFPAYLGFPED
VRNYFATNMGTSDPPTHTRLRKLVSQEFTVRRVEAMRPRVEQITAELLDEVGDSGVVDIVDRFAHPLPIKVICELLGVDE
KYRGEFGRWSSEILVMDPERAEQRGQAAREVVNFILDLVERRRTEPGDDLLSALIRVQDDDDGRLSADELTSIALVLLLA
GFESSVSLIGIGTYLLLTHPDQLALVRRDPSALPNAVEEILRYIAPPETTTRFAAEEVEIGGVAIPQYSTVLVANGAANR
DPKQFPDPHRFDVTRDTRGHLSFGQGIHFCMGRPLAKLEGEVALRALFGRFPALSLGIDADDVVWRRSLLLRGIDHLPVR
LDG


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