1jsv

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1jsv

The structure of cyclin-dependent kinase 2 (CDK2) in complex with 4-[(6-amino-4-pyrimidinyl)amino]benzenesulfonamide

Authors Clare, P.M. Poorman, R.A. Kelley, L.C. Watenpaugh, K.D. Bannow, C.A. Leach, K.L.
Citation The cyclin-dependent kinases cdk2 and cdk5 act by a random, anticooperative kinetic mechanism PubMed
Release date 2005-05-17
Exp. Method X-RAY DIFFRACTION
Resolution 1.96 Å
Classification TRANSFERASE

Sequence

Chain A (298 residues): Blast Uniprot EC 2.7.11.22
MENFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIRLDTETEGVPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVF
EFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFGVPVRTYT
HEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSF
PKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL


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