1k27
From PDBWiki
Crystal Structure of 5'-Deoxy-5'-Methylthioadenosine Phosphorylase in Complex with a Transition State Analogue
| Authors | Singh, V. Shi, W. Evans, G.B. Tyler, P.C. Furneaux, R.H. Almo, S.C. Schramm, V.L. |
| Citation | Picomolar transition state analogue inhibitors of human 5'-methylthioadenosine phosphorylase and X-ray structure with MT-immucillin-A PubMed |
| Release date | 2005-01-25 |
| Exp. Method | X-RAY DIFFRACTION |
| Resolution | 1.95 Å |
| Classification | TRANSFERASE |
Sequence
Chain A (283 residues): Blast Uniprot EC 2.4.2.28MASGTTTTAVKIGIIGGTGLDDPEILEGRTEKYVDTPFGKPSDALILGKIKNVDCVLLARHGRQHTIMPSKVNYQANIWA LKEEGCTHVIVTTACGSLREEIQPGDIVIIDQFIDRTTMRPQSFYDGSHSCARGVCHIPMAEPFCPKTREVLIETAKKLG LRCHSKGTMVTIEGPRFSSRAESFMFRTWGADVINMTTVPEVVLAKEAGICYASIAMATDYDCWKEHEEAVSVDRVLKTL KENANKAKSLLLTTIPQIGSTEWSETLHNLKNMAQFSVLLPRH
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| Databases | Visualization tools | Analysis tools | Quarternary structure |
|---|---|---|---|
Categories: K2 | PDB entry | X-RAY DIFFRACTION | TRANSFERASE | HOMO SAPIENS | 2005 | EC 2.4.2.28

