1klk

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1klk

CRYSTAL STRUCTURE OF PNEUMOCYSTIS CARINII DIHYDROFOLATE REDUCTASE TERNARY COMPLEX WITH PT653 AND NADPH

Authors Cody, V. Galitsky, N. Luft, J.R. Pangborn, W. Rosowsky, A. Queener, S.F.
Citation Structure-based enzyme inhibitor design: modeling studies and crystal structure analysis of Pneumocystis carinii dihydrofolate reductase ternary complex with PT653 and NADPH.
Release date 2002-12-12
Exp. Method X-RAY DIFFRACTION
Resolution 2.3 Å
Classification OXIDOREDUCTASE

Sequence

Chain A (206 residues): Blast Uniprot EC 1.5.1.3
MNQQKSLTLIVALTTSYGIGRSNSLPWKLKKEISYFKRVTSFVPTFDSFESMNVVLMGRKTWESIPLQFRPLKGRINVVI
TRNESLDLGNGIHSAKSLDHALELLYRTYGSESSVQINRIFVIGGAQLYKAAMDHPKLDRIMATIIYKDIHCDVFFPLKF
RDKEWSSVWKKEKHSDLESWVGTKVPHGKINEDGFDYEFEMWTRDL


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