1lqe

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1lqe

CRYSTAL STRUCTURE OF TRYPSIN IN COMPLEX WITH 79.

Authors Matter, H. Defossa, E. Heinelt, U. Blohm, P.M. Schneider, D. Mueller, A. Herok, S. Schreuder, H.A. Liesum, A. Brachvogel, V. Loenze, P. Walser, A. Al-Obeidi, F. Wildgoose, P.
Citation Design and quantitative structure-activity relationship of 3-amidinobenzyl-1H-indole-2-carboxamides

as potent, nonchiral, and selective inhibitors of blood coagulation factor Xa. PubMed

Release date 2004-01-13
Exp. Method X-RAY DIFFRACTION
Resolution 2.2 Å
Classification HYDROLASE

Sequence

Chain A (243 residues): Blast Uniprot EC 3.4.21.4
FIFLALLGAAVAFPVDDDDKIVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEG
NEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKA
PILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTI
ASN


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