1lqe
From PDBWiki
CRYSTAL STRUCTURE OF TRYPSIN IN COMPLEX WITH 79.
| Authors | Matter, H. Defossa, E. Heinelt, U. Blohm, P.M. Schneider, D. Mueller, A. Herok, S. Schreuder, H.A. Liesum, A. Brachvogel, V. Loenze, P. Walser, A. Al-Obeidi, F. Wildgoose, P. |
| Citation | Design and quantitative structure-activity relationship of 3-amidinobenzyl-1H-indole-2-carboxamides
as potent, nonchiral, and selective inhibitors of blood coagulation factor Xa. PubMed |
| Release date | 2004-01-13 |
| Exp. Method | X-RAY DIFFRACTION |
| Resolution | 2.2 Å |
| Classification | HYDROLASE |
Sequence
Chain A (243 residues): Blast Uniprot EC 3.4.21.4FIFLALLGAAVAFPVDDDDKIVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEG NEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKA PILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTI ASN
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| Databases | Visualization tools | Analysis tools | Quarternary structure |
|---|---|---|---|
Categories: LQ | PDB entry | X-RAY DIFFRACTION | HYDROLASE | 2004 | EC 3.4.21.4

