2b1z

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2b1z

Human estrogen receptor alpha ligand-binding domain in complex with 17methyl-17alpha-dihydroequilenin and a glucoc interacting protein 1 NR box II peptide

Authors Hsieh, R.W. Rajan, S.S. Sharma, S.K. Greene, G.L.
Citation Molecular characterization of a B-ring unsaturated estrogen: implications for conjugated equine estrogen components of premarin. PubMed
Release date 2006-09-19
Exp. Method X-RAY DIFFRACTION
Resolution 1.78 Å
Classification HORMONE/GROWTH FACTOR RECEPTOR

Sequence

Chain(s) C D (13 residues): Blast Uniprot
KHKILHRLLQDSS
Chain(s) A B (257 residues): Blast Uniprot
IKRSKKNSLALSLTADQMVSALLDAEPPILYSEYDPTRPFSEASMMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVH
LLEXAWLEILMIGLVWRSMEHPGKLLFAPNLLLDRNQGKXVEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSG
VYTFLSSTLKSLEEKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHLYSMKXKNVVPLS
DLLLEMLDAHRLHAPTS


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