2bmg
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CRYSTAL STRUCTURE OF FACTOR XA IN COMPLEX WITH 50
| Authors | Matter, H. Will, D.W. Nazare, M. Schreuder, H. Laux, V. Wehner, V. Liesum, A. |
| Citation | Structural Requirements for Factor Xa Inhibition by 3-Oxybenzamides with Neutral P1 Substituents: Combining X-Ray Crystallography, 3D-Qsar and Tailored Scoring Functions |
| Release date | 2006-03-08 |
| Exp. Method | X-RAY DIFFRACTION |
| Resolution | 2.7 Å |
| Classification | HYDROLASE |
Sequence
Chain A (53 residues): Blast Uniprot EC 3.4.21.6RKLCSLDNGDCDQFCHEEQNSVVCSCARGYTLADNGKACIPTGPYPCGKQTLEChain B (234 residues): Blast Uniprot EC 3.4.21.6
IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRF TKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSS SFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT
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| Databases | Visualization tools | Analysis tools | Quarternary structure |
|---|---|---|---|
Categories: BM | PDB entry | X-RAY DIFFRACTION | HYDROLASE | 2006 | EC 3.4.21.6

