2bmg

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2bmg

CRYSTAL STRUCTURE OF FACTOR XA IN COMPLEX WITH 50

Authors Matter, H. Will, D.W. Nazare, M. Schreuder, H. Laux, V. Wehner, V. Liesum, A.
Citation Structural Requirements for Factor Xa Inhibition by 3-Oxybenzamides with Neutral P1 Substituents: Combining X-Ray Crystallography, 3D-Qsar and Tailored Scoring Functions
Release date 2006-03-08
Exp. Method X-RAY DIFFRACTION
Resolution 2.7 Å
Classification HYDROLASE

Sequence

Chain A (53 residues): Blast Uniprot EC 3.4.21.6
RKLCSLDNGDCDQFCHEEQNSVVCSCARGYTLADNGKACIPTGPYPCGKQTLE
Chain B (234 residues): Blast Uniprot EC 3.4.21.6
IVGGQECKDGECPWQALLINEENEGFCGGTILSEFYILTAAHCLYQAKRFKVRVGDRNTEQEEGGEAVHEVEVVIKHNRF
TKETYDFDIAVLRLKTPITFRMNVAPACLPERDWAESTLMTQKTGIVSGFGRTHEKGRQSTRLKMLEVPYVDRNSCKLSS
SFIITQNMFCAGYDTKQEDACQGDSGGPHVTRFKDTYFVTGIVSWGEGCARKGKYGIYTKVTAFLKWIDRSMKT


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