2cn8

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2cn8

CRYSTAL STRUCTURE OF HUMAN CHK2 IN COMPLEX WITH DEBROMOHYMENIALDISINE

Authors Oliver, A.W. Paul, A. Boxall, K.J. Barrie, S.E. Aherne, G.W. Garrett, M.D. Mittnacht, S. Pearl, L.H.
Citation Trans-activation of the DNA-damage signalling protein kinase Chk2 by T-loop exchange. PubMed
Release date 2007-01-03
Exp. Method X-RAY DIFFRACTION
Resolution 2.7 Å
Classification TRANSFERASE

Sequence

Chain A (329 residues): Blast Uniprot EC 2.7.11.1
GPLGSHMSVYPKALRDEYIMSKTLGSGACGEVKLAFERKTCKKVAIKIISKRKFAIGSAREADPALNVETEIEILKKLNH
PCIIKIKNFFDAEDYYIVLELMEGGELFDKVVGNKRLKEATCKLYFYQMLLAVQYLHENGIIHRDLKPENVLLSSQEEDC
LIKITDFGHSKILGETSLMRTLCGTPTYLAPEVLVSVGTAGYNRAVDCWSLGVILFICLSGYPPFSEHRTQVSLKDQITS
GKYNFIPEVWAEVSEKALDLVKKLLVVDPKARFTTEEALRHPWLQDEDMKRKFQDLLSEENESTALPQVLAQPSTSRKRP
REGEAEGAE


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