2csn

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2csn

BINARY COMPLEX OF CASEIN KINASE-1 WITH CKI7

Authors Xu, R.M. Carmel, G. Kuret, J. Cheng, X.
Citation Structural basis for selectivity of the isoquinoline sulfonamide family of protein kinase inhibitors.
Release date 1996-03-08
Exp. Method X-RAY DIFFRACTION
Resolution 2.5 Å
Classification PROTEIN KINASE

Sequence

Chain A (297 residues): Blast Uniprot EC 2.7.11.1
SGQNNVVGVHYKVGRRIGEGSFGVIFEGTNLLNNQQVAIKFEPRRSDAPQLRDEYRTYKLLAGCTGIPNVYYFGQEGLHN
VLVIDLLGPSLEDLLDLCGRKFSVKTVAMAAKQMLARVQSIHEKSLVYRDIKPDNFLIGRPNSKNANMIYVVDFGMVKFY
RDPVTKQHIPYREKKNLSGTARYMSINTHLGREQSRRDDLEALGHVFMYFLRGSLPWQGLKAATNKQKYERIGEKKQSTP
LRELCAGFPEEFYKYMHYARNLAFDATPDYDYLQGLFSKVLERLNTTEDENFDWNLL


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