2jbo

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2jbo

PROTEIN KINASE MK2 IN COMPLEX WITH AN INHIBITOR (CRYSTAL FORM-1, SOAKING)

Authors Hillig, R.C. Eberspaecher, U. Monteclaro, F. Huber, M. Nguyen, D. Mengel, A. Muller-Tiemann, B. Egner, U.
Citation Structural Basis for a High Affinity Inhibitor Bound to Protein Kinase Mk2.
Release date 2008-01-08
Exp. Method X-RAY DIFFRACTION
Resolution 3.1 Å
Classification TRANSFERASE

Sequence

Chain A (326 residues): Blast Uniprot
GSQQFPQFHVKSGLQIKKNAIIDDYKVTSQVLGLGINGKVLQIFNKRTQEKFALKMLQDCPKARREVELHWRASQCPHIV
RIVDVYENLYAGRKCLLIVMECLDGGELFSRIQDRGDQAFTEREASEIMKSIGEAIQYLHSINIAHRDVKPENLLYTSKR
PNAILKLTDFGFAKETTSHNSLTTPCYTPYYVAPEVLGPEKYDKSCDMWSLGVIMYILLCGYPPFYSNHGLAISPGMKTR
IRMGQYEFPNPEWSEVSEEVKMLIRNLLKTEPTQRMTITEFMNHPWIMQSTKVPQTPLHTSRVLKEDKERWEDVKEEMTS
ALATMR


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