2p3g
From PDBWiki
Crystal structure of a pyrrolopyridine inhibitor bound to MAPKAP Kinase-2
| Authors | Anderson, D.R. Meyers, M.J. Vernier, W.F. Mahoney, M.W. Kurumbail, R.G. Caspers, N. Poda, G.I. Schindler, J.F. Reitz, D.B. Mourey, R.J. |
| Citation | Pyrrolopyridine Inhibitors of Mitogen-Activated Protein Kinase-Activated Protein Kinase 2 (MK-2). PubMed |
| Release date | 2007-06-12 |
| Exp. Method | X-RAY DIFFRACTION |
| Resolution | 3.8 Å |
| Classification | TRANSFERASE |
Sequence
Chain X (327 residues): Blast Uniprot EC 2.7.11.1QFHVKSGLQIKKNAIIDDYKVTSQVLGLGINGKVLQIFNKRTQEKFALKMLQDCPKARREVELHWRASQCPHIVRIVDVY ENLYAGRKCLLIVMECLDGGELFSRIQDRGDQAFTEREASEIMKSIGEAIQYLHSINIAHRDVKPENLLYTSKRPNAILK LTDFGFAKETTSHNSLTTPCYTPYYVAPEVLGPEKYDKSCDMWSLGVIMYILLCGYPPFYSNHGLAISPGMKTRIRMGQY EFPNPEWSEVSEEVKMLIRNLLKTEPTQRMTITEFMNHPWIMQSTKVPQTPLHTSRVLKEDKERWEDVKEEMTSALATMR VDYEQIK
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