2p3g

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2p3g

Crystal structure of a pyrrolopyridine inhibitor bound to MAPKAP Kinase-2

Authors Anderson, D.R. Meyers, M.J. Vernier, W.F. Mahoney, M.W. Kurumbail, R.G. Caspers, N. Poda, G.I. Schindler, J.F. Reitz, D.B. Mourey, R.J.
Citation Pyrrolopyridine Inhibitors of Mitogen-Activated Protein Kinase-Activated Protein Kinase 2 (MK-2). PubMed
Release date 2007-06-12
Exp. Method X-RAY DIFFRACTION
Resolution 3.8 Å
Classification TRANSFERASE

Sequence

Chain X (327 residues): Blast Uniprot EC 2.7.11.1
QFHVKSGLQIKKNAIIDDYKVTSQVLGLGINGKVLQIFNKRTQEKFALKMLQDCPKARREVELHWRASQCPHIVRIVDVY
ENLYAGRKCLLIVMECLDGGELFSRIQDRGDQAFTEREASEIMKSIGEAIQYLHSINIAHRDVKPENLLYTSKRPNAILK
LTDFGFAKETTSHNSLTTPCYTPYYVAPEVLGPEKYDKSCDMWSLGVIMYILLCGYPPFYSNHGLAISPGMKTRIRMGQY
EFPNPEWSEVSEEVKMLIRNLLKTEPTQRMTITEFMNHPWIMQSTKVPQTPLHTSRVLKEDKERWEDVKEEMTSALATMR
VDYEQIK


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