2pdx

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2pdx

Human aldose reductase double mutant S302R-C303D complexed with zopolrestat.

Authors Steuber, H. Heine, A. Podjarny, A. Klebe, G.
Citation Merging the binding sites of aldose and aldehyde reductase for detection of inhibitor selectivity-determining features. PubMed
Release date 2008-04-01
Exp. Method X-RAY DIFFRACTION
Resolution 1.65 Å
Classification OXIDOREDUCTASE

Sequence

Chain(s) A (316 residues): Blast Uniprot EC 1.1.1.21
MASRILLNNGAKMPILGLGTWKSPPGQVTEAVKVAIDVGYRHIDCAHVYQNENEVGVAIQEKLREQVVKREELFIVSKLW
CTYHEKGLVKGACQKTLSDLKLDYLDLYLIHWPTGFKPGKEFFPLDESGNVVPSDTNILDTWAAMEELVDEGLVKAIGIS
NFNHLQVEMILNKPGLKYKPAVNQIECHPYLTQEKLIQYCQSKGIVVTAYSPLGSPDRPWAKPEDPSLLEDPRIKAIAAK
HNKTTAQVLIRFPMQRNLVVIPKSVTPERIAENFKVFDFELSSQDMTTLLSYNRNWRVCALLRDTSHKDYPFHEEF

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