2rjq

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2rjq

Crystal structure of ADAMTS5 with inhibitor bound

Authors Mosyak, L. Georgiadis, K. Shane, T. Svenson, K. Hebert, T. McDonagh, T. Mackie, S. Olland, S. Lin, L. Zhong, X. Kriz, R. Reifenberg, E.L. Collins-Racie, L.A. Corcoran, C. Freeman, B. Zollner, R. Marvell, T. Vera, M. Sum, P.E. Lavallie, E.R. Stahl, M. Somers, W.
Citation Crystal structures of the two major aggrecan degrading enzymes, ADAMTS4 and ADAMTS5. PubMed
Release date 2008-01-08
Exp. Method X-RAY DIFFRACTION
Resolution 2.6 Å
Classification HYDROLASE

Sequence

Chain A (378 residues): Blast Uniprot EC 3.4.24.-
SISRARQVELLLVADASMARLYGRGLQHYLLTLASIANRLYSHASIENHIRLAVVKVVVLGDKDKSLEVSKNAATTLKNF
CKWQHQHNQLGDDHEEHYDAAILFTREDLCGHHSCDTLGMADVGTICSPERSCAVIEDDGLHAAFTVAHEIGHLLGLSHD
DSKFCEETFGSTEDKRLMSSILTSIDASKPWSKCTSATITEFLDDGHGNCLLDLPRKQILGPEELPGQTYDATQQCNLTF
GPEYSVCPGMDVCARLWCAVVRQGQMVCLTKKLPAVEGTPCGKGRICLQGKCVDKTKKKYYSTSSHGNWGSWGSWGQCSR
SCGGGVQFAYRHCNNPAPRNNGRYCTGKRAIYRSCSLMPCPPNGKSFGSAWSHPQFEK


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