3bgs

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3bgs

Structure of human purine nucleoside phosphorylase with L-DADMe-ImmH and phosphate

Authors Rinaldo-Matthis, A. Murkin, A.S. Ramagopal, U.A. Clinch, K. Mee, S.P. Evans, G.B. Tyler, P.C. Furneaux, R.H. Almo, S.C. Schramm, V.L.
Citation L-Enantiomers of transition state analogue inhibitors bound to human purine nucleoside phosphorylase PubMed
Release date 2008-02-26
Exp. Method X-RAY DIFFRACTION
Resolution 2.099 Å
Classification TRANSFERASE

Sequence

Chain A (289 residues): Blast Uniprot EC 2.4.2.1
MENGYTYEDYKNTAEWLLSHTKHRPQVAIICGSGLGGLTDKLTQAQIFDYSEIPNFPRSTVPGHAGRLVFGFLNGRACVM
MQGRFHMYEGYPLWKVTFPVRVFHLLGVDTLVVTNAAGGLNPKFEVGDIMLIRDHINLPGFSGQNPLRGPNDERFGDRFP
AMSDAYDRTMRQRALSTWKQMGEQRELQEGTYVMVAGPSFETVAECRVLQKLGADAVGMSTVPEVIVARHCGLRVFGFSL
ITNKVIMDYESLEKANHEEVLAAGKQAAQKLEQFVSILMASIPLPDKAS


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