3bm8

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3bm8

crystal structure of YopH mutant D356A complexed with irreversible inhibitor PVSN

Authors Liu, S. Zhou, B. Yang, H. He, Y. Jiang, Z.X. Kumar, S. Wu, L. Zhang, Z.Y.
Citation Aryl vinyl sulfonates and sulfones as active site-directed and mechanism-based probes for protein tyrosine phosphatases. PubMed
Release date 2008-06-17
Exp. Method X-RAY DIFFRACTION
Resolution 2.7 Å
Classification HYDROLASE

Sequence

Chain(s) A (305 residues): Blast Uniprot EC 3.1.3.48
RERPHTSGHHGAGEARATAPSTVSPYGPEARAELSSRLTTLRNTLAPATNDPRYLQACGGEKLNRFRDIQCRRQTAVRAD
LNANYIQVGNTRTIACQYPLQSQLESHFRMLAENRTPVLAVLASSSEIANQRFGMPDYFRQSGTYGSITVESKMTQQVGL
GDGIMADMYTLTIREAGQKTISVPVVHVGNWPAQTAVSSEVTKALASLVDQTAETKRNMYESKGSSAVADDSKLRPVIHC
RAGVGRTAQLIGAMCMNDSRNSQLSVEDMVSQMRVQRNGIMVQKDEQLDVLIKLAEGQGRPLLNS

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