3bm8
From PDBWiki
crystal structure of YopH mutant D356A complexed with irreversible inhibitor PVSN
| Authors | Liu, S. Zhou, B. Yang, H. He, Y. Jiang, Z.X. Kumar, S. Wu, L. Zhang, Z.Y. |
| Citation | Aryl vinyl sulfonates and sulfones as active site-directed and mechanism-based probes for protein tyrosine phosphatases. PubMed |
| Release date | 2008-06-17 |
| Exp. Method | X-RAY DIFFRACTION |
| Resolution | 2.7 Å |
| Classification | HYDROLASE |
Sequence
Chain(s) A (305 residues): Blast Uniprot EC 3.1.3.48RERPHTSGHHGAGEARATAPSTVSPYGPEARAELSSRLTTLRNTLAPATNDPRYLQACGGEKLNRFRDIQCRRQTAVRAD LNANYIQVGNTRTIACQYPLQSQLESHFRMLAENRTPVLAVLASSSEIANQRFGMPDYFRQSGTYGSITVESKMTQQVGL GDGIMADMYTLTIREAGQKTISVPVVHVGNWPAQTAVSSEVTKALASLVDQTAETKRNMYESKGSSAVADDSKLRPVIHC RAGVGRTAQLIGAMCMNDSRNSQLSVEDMVSQMRVQRNGIMVQKDEQLDVLIKLAEGQGRPLLNS
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