3bmy
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Discovery of Benzisoxazoles as Potent Inhibitors of Chaperone Hsp90
| Authors | Gopalsamy, A. Shi, M. Golas, J. Vogan, E. Jacob, J. Johnson, M. Lee, F. Nilakantan, R. Petersen, R. Svenson, K. Chopra, R. Tam, M.S. Wen, Y. Ellingboe, J. Arndt, K. Boschelli, F. |
| Citation | Discovery of benzisoxazoles as potent inhibitors of chaperone heat shock protein 90. PubMed |
| Release date | 2008-07-08 |
| Exp. Method | X-RAY DIFFRACTION |
| Resolution | 1.6 Å |
| Classification | Chaperone |
Sequence
Chain(s) A (226 residues): Blast UniprotQPMEEEVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLT IVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSF TVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEKERDKEVSDDEAE
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| Databases | Visualization tools | Analysis tools | Quarternary structure |
|---|---|---|---|
Categories: BM | PDB entry | X-RAY DIFFRACTION | CHAPERONE | HOMO SAPIENS | 2008

