3tgk

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3tgk

TRYPSINOGEN MUTANT D194N AND DELETION OF ILE 16-VAL 17 COMPLEXED WITH BOVINE PANCREATIC TRYPSIN INHIBITOR (BPTI)

Authors Pasternak, A. White, A. Jeffery, C.J. Medina, N. Cahoon, M. Ringe, D. Hedstrom, L.
Citation The energetic cost of induced fit catalysis: Crystal structures of trypsinogen mutants with enhanced activity and inhibitor affinity. PubMed
Release date 2001-07-04
Exp. Method X-RAY DIFFRACTION
Resolution 1.7 Å
Classification HYDROLASE/ HYDROLASE INHIBITOR

Sequence

Chain E (231 residues): Blast Uniprot EC 3.4.21.4
EAFPVDDDDKGGYTCQENSVPYQVSLNSGYHFCGGSLINDQWVVSAAHCYKSRIQVRLGEHNINVLEGNEQFVNAAKIIK
HPNFDRKTLNNDIMLIKLSSPVKLNARVATVALPSSCAPAGTQCLISGWGNTLSSGVNEPDLLQCLDAPLLPQADCEASY
PGKITDNMVCVGFLEGGKDSCQGNSGGPVVCNGELQGIVSWGYGCALPDNPGVYTKVCNYVDWIQDTIAAN
Chain I (65 residues): Blast Uniprot
RPDFCLEPPYTGPCKARIIRYFYNAKAGLCQTFVYGGCRAKRNNFKSAEDCMRTCGGAIGPWENL


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